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Brightening

Tranexamic Acid

One of the new stars in the fight against hyperpigmentation — tranexamic acid blocks melanin at a different stage than vitamin C or arbutin, and is well tolerated even by sensitive skin. Effective against melasma and post-acne spots.

anti-pigmentationmelasmabrighteningsensitive skin
✓ Safe
Comedogenic Rating
0/5
Irritation Potential
0/5

What is it?

Tranexamic acid (TXA) — a synthetic derivative of the amino acid lysine. Initially developed as an anticoagulant in medicine. In INCI: Tranexamic Acid. It blocks the interaction of plasmin with keratinocytes, reducing the release of arachidonic acid and stimulating melanocytes. The mechanism of action differs from tyrosinase inhibitors — it can synergistically combine with them.

Brightening active in targeted serums for melasma, post-inflammatory pigmentation, and uneven skin tone. Especially effective for hormone-induced hyperpigmentation (melasma) — a problem where classic remedies are often insufficient.

Key Benefits

✦
Effective treatment for melasma
TXA blocks plasmin-induced stimulation of melanocytes — especially effective for melasma (hormonal pigmentation), where other products are less effective. Clinical studies show comparable or higher efficacy than kojic acid and azelaic acid.
◈
Gentle tolerance profile
Not an acid in the classical sense — does not lower the pH of the formula, does not irritate the skin. Ideal for sensitive skin and for those who cannot tolerate traditional brightening acids.
✧
Synergy with other brightening agents
Since TXA blocks a different pathway of melanogenesis (plasmin) than tyrosinase inhibitors (vitamin C, niacinamide, arbutin) — the combination yields an effect that significantly exceeds the sum of its parts.

Suitable for

skin with melasmaskin with post-acne spotssensitive skinall skin types

Main Actions

✓ reduction of melasma✓ brightening of pigmented spots✓ evening out skin tone
Time is needed for results

Tranexamic acid works slower than acid brightening agents — noticeable results at 2–5% concentration appear after 8–12 weeks of regular use. Do not expect an instant effect — this is a marathon product for sustainable results.

CategoryBrightening
From our blog
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Frequently Asked Questions

What does Tranexamic Acid do for skin?
Brightening active in targeted serums for melasma, post-inflammatory pigmentation, and uneven skin tone. Especially effective for hormone-induced hyperpigmentation (melasma) — a problem where classic remedies are often insufficient.
Who should use Tranexamic Acid?
Tranexamic Acid is suitable for: skin with melasma, skin with post-acne spots, sensitive skin, all skin types.
Are there any warnings about Tranexamic Acid?
Tranexamic acid works slower than acid brightening agents — noticeable results at 2–5% concentration appear after 8–12 weeks of regular use. Do not expect an instant effect — this is a marathon product for sustainable results.

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